Introduction to biopharmaceutics, study on process evolved after drug administration: absorption, distribution, metabolism and elimination in human and animals including effects of drug delivery systems on these processes; factors affecting drug bioavailability, biopharmaceutical classification systems, pharmacokinetic calculations, pharmacokinetic parameters, pharmacokinetic compartment models; application of pharmacokinetics/ pharmacodynamics/ biopharmaceutics concepts in drug design, drug delivery systems; bioequivalence study, drug and delivery selection.